Adenosine 3',5'-cyclic Monophosphorothioate, Rp-Isomer, Triethylammonium Salt-CAS 151837-09-1-Calbiochem

C₁₀H₁₁N₅O₅PS · 4C₆H₁₆N

753.06

Note: 5 µmol = 2.23 mg.
A cell-permeable and reversible inhibitor of protein kinase A (K_i = 11 µM). Resistant to hydrolysis by phosphodiesterases. Noncompetitive with respect to ATP.
Cell permeable inhibitor of protein kinase A (K_i = 11 µM). Resistant to hydrolysis by phosphodiesterases. Note: 5 µmol = 2.23 mg

Cell permeable: yes
Product does not compete with ATP.
Target K_i: 11 µM against protein kinase A
Reversible: yes
Primary Target
PKA

Toxicity: Standard Handling (A)

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.

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Dostmann, W.R., et al. 1990. J. Biol. Chem.265, 10484.
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Eckstein, F. 1985. Annu. Rev. Biochem.54, 367.
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O′Brian, C.A., et al. 1982. Biochemistry21, 4371.

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

100

≥98% (HPLC)

crystalline solid

Calbiochem^®

OK to freeze
desiccated (hygroscopic)

water: 20 mg/mL

wet ice

−20℃

5 μmol in Glass bottle

11 - Combustible Solids

WGK 2